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active-site directed and substrate competitive AKR1C1 inhibitor (Ki = 4 nM) with moderate to excellent selectivity over AKR1C2
but TSC1+/+ cells are resistant
Dissolve 0
CN1[C@@H]2C[C@@H](O)C[C@H]1[C@@H]1O[C@H]21
Solubility: DMSO: 56 mg/mL(201
Telotristat 845 active-site directed and substrate competitiveTelotristat, also known as LP 778902, is the acid form of Telotristat ethyl, and the active metabolite of LX1606 (Telotristat etiprate), which is an orally bioavailable, small molecule, tryptophan hydroxylase (TPH) inhibitor and serotonin synthesis inhibitor with potential antiserotonergic activity. Blocking peripheral serotonin synthesis by telotristat reduces severity of both chemical and infection induced intestinal inflammation. Product
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